Bldg.12 1233
[Organic Chemistry -Reaction and Synthesis- Heterocyclic Compounds]
Thursday, March 26, AM
Chair: MUTOH, Yuichiro
(09:00-10:00)
* 8:50-9:00: interval for laptop PC connection.(1G3-01, 1G3-02, 1G3-03, 1G3-04, 1G3-05)
1G3-01
Photochemical Reactions of 1,3-diphenyltetrazolium-5-thiolates with an isopropyl group or ethnyl group at the ortho position (Grad Sch. Eng., Nagoya Inst. of Tech.) º DOI, Akihiro; YAMASHITA, Yukinobu; HIRASHITA, Tsunehisa; ARAKI, Shuki
1G3-02
Reactions of 1,3-diphenyltetrazolium-5-hydroxylamide (Grad Sch. Eng., Nagoya Inst. of Tech.) º MATSUKAWA, Yuta; HIRASHITA, Tsunehisa; ARAKI, Shuki
1G3-03
Nucleophilic Addition of Tetrazoles to Haloalkynes and Its Application (Grad. Sch. Biosci. Biotech., Tokyo Tech) YAMAGISHI, Masahito; º KOYANAGI, Tetsuya; HATA, Takeshi; URABE, Hirokazu
1G3-04
Cyclization Reaction of Substituted Alkenyl Esters and Amides of Ethenetricarboxylate (Nara Univ. of Educ.; Grad. Sch. Mat. Sci., NAIST) YAMAZAKI, Shoko; º WADA, Junya; KAKIUCHI, Kiyomi
1G3-05*
Synthesis of α-functionalized unsaturated oximes and heterocyclic compounds by Umpolung substitution using nitrosoallenes (Grad. Sch. Mat. Sci., NAIST) º TANIMOTO, Hiroki; MIZUTANI, Yusuke; YOKOYAMA, Keiichi; KAKIUCHI, Kiyomi
Chair: TANIMOTO, Hiroki
(10:10-11:10)
* 10:00-10:10: interval for laptop PC connection.(1G3-08, 1G3-09, 1G3-10, 1G3-11, 1G3-12, 1G3-13)
1G3-08
Catalytic Cyclization of Allyl Amides of Ethenetricarboxylate Promoted by Lewis acid (Nara Univ. of Educ.; Grad. Sch. Mat. Sci., NAIST) YAMAZAKI, Shoko; º NIINA, Mamiko; KAKIUCHI, Kiyomi
1G3-09
Copper(II)-Catalyzed [4+1] Annulation of Propargylamines with N,O-Acetals: New Entry to Synthesis of Polysubstituted Pyrrole Derivatives (Fac. Sci. Technol., Tokyo Univ. of Sci.) º HORI, Hiroaki; OGIWARA, Yohei; SAKAI, Norio
1G3-10
Indium-Catalyzed One-pot Preparation of N-Substituted Lactams via Direct Reductive Amination of Keto Acids with Primary Amines (Fac. Sci. Technol., Tokyo Univ. of Sci.) º UCHIYAMA, Takuya; OGIWARA, Yohei; SAKAI, Norio
1G3-11
Synthesis of multiply substituted piperidines based on Cu-catalyzed formation of 1,6-dihydropyridines (Grad. Sch. Chi Sci. and Eng., Hokkaido Univ.; Fac. Sci., Hokkaido Univ.) º WATANABE, Ryo; MIZOGUCHI, Haruki; MINAMI, Shintaro; OGURI, Hiroki; OIKAWA, Hideaki
1G3-12
A Short-Step Construction of Fused Pyridine Alkaloid Skeletons via a Key Step involving Hetero Diels-Alder Reaction of Isotellurazoles (Grad. Sch. Eng., Iwate Univ.) SHIMADA, Kazuaki; º TANEICHI, Yusuke; KORENAGA, Toshinobu
1G3-13
Compounds having imidazo[1,5-a]pyridine skeleton with organometallic reagents (Chubu Univ. Department of Applied Chemistry, College of Engineering) º KAMIYA, Kenji; KUSUNOSE, Masashi; NIYOMURA, Osamu
Chair: YAMAZAKI, Shoko
(11:20-12:20)
* 11:10-11:20: interval for laptop PC connection.(1G3-15, 1G3-16, 1G3-18, 1G3-19, 1G3-20)
1G3-15
Chromium Oxide-Catalyzed Oxidation of Dimethyl- and Diethyl-2,2'-bipyridines (TITC Central Research Institute) º YAMAZAKI, Shigekazu
1G3-16*
Synthesis of N,N,2,6-Tetrasubstituted 4-Nitroalinines by Three Component Ring Transformation of Dinitropyridone (Sch. Env. Sci. Eng., KUT) º LE, Thi Song; ASAHARA, Haruyasu; NISHIWAKI, Nagatoshi
1G3-18
Synthesis of 3,5-Dinitro-1,4-dihydropyridines by the Condensation of Formylnitroenamine with Aldehydes (Sch. Env. Sci. Eng., KUT) º HAMADA, Mai; ASAHARA, Haruyasu; NAKAIKE, Yumi; NISHIWAKI, Nagatoshi
1G3-19
Effective Skeletal Construction of 4-aminopyrimidines and 4-aminoquinazolines with β-cyanoenamines and isocyanides (Fac. Sci. Technol., Tokyo Univ. of Sci.) º NAKANO, Tsukasa; KATO, Takubo; OGIWARA, Yohei; SAKAI, Norio; KONAKAHARA, Takeo
1G3-20
NHC-catalyzed nucleophilic aroylation of quinazoline at the C5-C8 position (Grad. Sch. of Sci. Technol., Sophia Univ.) º NAKAGAWA, Mizuki; SUZUKI, Yumiko
Thursday, March 26, PM
Chair: YAMAGUCHI, Eiji
(13:30-14:30)
* 13:20-13:30: interval for laptop PC connection.(1G3-28, 1G3-29, 1G3-30, 1G3-31, 1G3-32)
1G3-28
Acid-promoted Intramolecular Hetero Diels-Alder Reaction of o-Alkynylphenylcarbodiimide (Fac. Sci., Tokyo Univ. of Sci.; Univ. of Tsukuba International Institute for Integrative Sleep Medicine) º KOYAMA, Yasuaki; KUTSUMURA, Noriki; NAGASE, Hiroshi; SAITO, Takao
1G3-29
Catalytic Synthesis of Isoquinoline Derivatives from Imines through Migration of Substituents on Nitrogen (Grad. Sch. Eng., Osaka Univ.) º SASAOKA, Yukari; HOSHIMOTO, Yoichi; OHASHI, Masato; OGOSHI, Sensuke
1G3-30
Development of the Pd(II)-catalyzed cyclization and its application to the synthetic studies of carbazole alkaloids (Univ. of Toyama ,Graduate school of science and engineering) YOKOYAMA, Hajime; º SHOJI, Yuzen; KUBO, Takayoshi; MATSUMURA, Yosuke; HOSOKAWA, Junichi; MIYAZAWA, Masahiro; HIRAI, Yoshiro
1G3-31
Synthesis of tricyclic benzazonines by the acid-catalyzed aza-Prins reaction (Fac. Sci., Tokyo Univ. of Sci.) º KATAMURA, Tomohiro; SHIMIZU, Tomoaki; MUTOH, Yuichiro; SAITO, Shinichi
1G3-32*
Functionalization of the 1-Methyl-2-quinolone Framework Activated by Steric Repulsion of the Substituents (Sch. Env. Sci. Eng., KUT) ASAHARA, Haruyasu; CHEN, Xin; º NISHIWAKI, Nagatoshi
Chair: NISHIWAKI, Nagatoshi
(14:40-15:40)
* 14:30-14:40: interval for laptop PC connection.(1G3-35, 1G3-36, 1G3-38, 1G3-39, 1G3-40)
1G3-35
Novel synthesis of isoindoles using pyrolysis reaction (Grad. Sch. Eng., Utsunomiya Univ.) º SHINOZAKI, Yasutaka; OBA, Toru; ITO, Naotsugu; SATO, Takafumi; ITO, Satoshi
1G3-36*
Synthesis of 3,4-fused 2-quinolones from (o-aminophenyl)propiolate via cycloaddition (Grad. Sch. Pharm. Sci., Nagoya Univ.) º MURAYAMA, Tsukasa; SHIBUYA, Masatoshi; YAMAMOTO, Yoshihiko
1G3-38
Development of synthetic method toward polycyclic heterocycles by means of visible right mediated radical cyclization (Gifu Pharm. Univ.) º SUDO, Yusuke; YAMAGUCHI, Eiji; TADA, Norihiro; ITOH, Akichika
1G3-39
Synthesis of novel Spiro [indole-pyrazoles] using isocyanide based multi component reaction (Grad. Sch. Eng., KIT) º JALLI, Venkataprasad; MORIGUCHI, Tetsuji; ARAKI, Koji; TSUGE, Akihiko
1G3-40
Phosphinic acid-promoted addition reaction of isocyanides to 1-methoxyisochroman (Grad. Sch. Nat. Sci. Technol., Kanazawa Univ.) º MATSUZAKI, Syunsuke; SOETA, Takahiro; UKAJI, Yutaka
Chair: YAMAMOTO, Yoshihiko
(15:50-16:40)
* 15:40-15:50: interval for laptop PC connection.(1G3-42, 1G3-44, 1G3-45, 1G3-46)
1G3-42*
Intramolecular C-H Amination of Aromatic Compounds via Electron Transfer (Grad. Sch. Eng., Kyoto Univ.) º MOROFUJI, Tatsuya; SHIMIZU, Akihiro; YOSHIDA, Jun-ichi
1G3-44
Intramolecular cyclization of 2-(N-pyrrolylsulfenyl)benzoic acid (IRC3, AIST; Fac. Sci. Technol., Tokyo Univ. of Sci.) SHIMIZU, Masao; º MASUDA, Kotaro; TANAKA, Shinji; ANDO, Wataru; SAKAI, Norio
1G3-45
Synthesis of Various 1,3-Thiazole Derivatives through Oxidative Ring Closure of 1,3-Thiaza-1,3-butadienes (Grad. Sch. Eng., Iwate Univ.) SHIMADA, Kazuaki; º ISOGAMI, Megumi; KORENAGA, Toshinobu
1G3-46
Substituent Effect on Ring-expansion Reaction of Vinylsulfonium Ylide (Kobe City Coll. Technol.) º ICHINOSE, Yuma; KOIZUMI, Takuya
Friday, March 27, AM
Chair: SENGOKU, Tetsuya
(09:00-10:00)
* 8:50-9:00: interval for laptop PC connection.(2G3-01, 2G3-02, 2G3-03, 2G3-04, 2G3-05, 2G3-06)
2G3-01
Mn(III)-Based Oxidation of 3-Ethenyl-2,4-pentanediones and their Derivatives (Grad. Sch. Sci. Technol., Kumamoto Univ.) º HASHIMOTO, Shintarou; NISHINO, Hiroshi
2G3-02
Oxazolidine synthesis by three component reaction of diazo compound, aldehyde, and imine-Scope and limitation of substrates (Grad. Sch. Sci. Technol., Shinshu Univ.) º KAMIYA, Hideaki; SUGA, Hiroyuki
2G3-03
Palladium-catalyzed Dipolar Cycloaddition Reactions of Oxidopyrylium Ylides with Olefinic Dipolarophiles (Grad. Sch. Sci. Technol., Shinshu Univ.) º TAKAHASHI, Kie; KIMURA, Miyuki; IWAI, Taichi; SUGA, Hiroyuki
2G3-04
Development of the synthetic method of furoxan derivatives (Grad. Sch. Sci., Kobe Univ.) º ANDO, Akihiro; MATSUBARA, Ryosuke
2G3-05
Withdrawn
2G3-06
Preparation of Oxazoles from Ketones and Nitriles with Molecular Iodine and Oxone (Grad. Sch. Sci., Chiba Univ.) º IMAI, Sho; MORIYAMA, Katsuhiko; TOGO, Hideo
Chair: YOSHIMATSU, Mitsuhiro
(10:10-11:10)
* 10:00-10:10: interval for laptop PC connection.(2G3-08, 2G3-09, 2G3-10, 2G3-11, 2G3-12, 2G3-13)
2G3-08
Synthesis of lamellarins using [1]benzopyrano[3,4-b]pyrrol-4(3H)-one as a key intermediate (1) (Grad. Sch. Eng., Nagasaki Univ.) º KATAE, Takatoshi; HARADA, Issei; FUKUDA, Tsutomu; IWAO, Masatomo
2G3-09
Synthesis of lamellarins using [1]benzopyrano[3,4-b]pyrrol-4(3H)-one as a key intermediate (2) (Grad. Sch. Eng., Nagasaki Univ.) º HARADA, Issei; KATAE, Takatoshi; FUKUDA, Tsutomu; IWAO, Masatomo
2G3-10
Synthesis of 6-halogenated lamellarin N derivatives (Grad. Sch. Eng., Nagasaki Univ.) º TOKUSHIMA, Keiji; FUKUDA, Tsutomu; IWAO, Masatomo
2G3-11
Total Synthesis of Clavicipitic Acid via Ir-Catalyzed C-H Bond Activation (Sch. Advanced Sci. Eng., Waseda Univ.) º ITO, Mamoru; TAHARA, Yu-ki; SHIBATA, Takanori
2G3-12
Development of Stereoselective Synthesis of Marinolic Acid A, An Anti-MRSA Agent (Grad. Sch. Eng., Shizuoka Univ.) SENGOKU, Tetsuya; º MOMOSE, Naoto; WARASINA, Takuya; TAKAHASHI, Masaki; YODA, Hidemi
2G3-13
Chichibabin pyridine synthesis of the COPD biomarker isodesmosine (Fac. Sci., Sophia Univ.) º KOMATSU, Akira; SUGIMURA, Takanori; TANIGAWA, Takahiro; KOSEKI, Yohei; USUKI, Toyonobu
Chair: SUZUKI, Yumiko
(11:20-12:20)
* 11:10-11:20: interval for laptop PC connection.(2G3-15, 2G3-16, 2G3-17, 2G3-18, 2G3-19, 2G3-20)
2G3-15
Synthesis of benzofuropyrazoles as a new class of hypoxia inducible factor (HIF)-1 inhibitors. (Grad. Sch. Sci. and Technol., Gakushuin Univ.) º MINEGISHI, Hidemitsu; NAKAMURA, Hiroyuki
2G3-16
Nucleic Base-Promoted Cyclization of 1,6-Diynes (Fac. Edu., Gifu Univ.) º KOBAYASHI, Yuka; YOSHIMATSU, Mitsuhiro
2G3-17
Rhodium-catalyzed synthesis of benzo naphthopyranone from diazonaphthoquinone (Grad. Sch. Eng., KIT) º TAKAHASHI, Shuhei; KANEMURA, Koichi; OKAUCHI, Tatsuo; KITAMURA, Mitsuru
2G3-18
Synthesis of Aryl Azides from phenol with guanidino diazonium salt (Grad. Sch. Eng., KIT) º MURAKAMI, Kento; KOGA, Tatsuya; OKAUCHI, Tatsuo; KITAMURA, Mitsuru
2G3-19
The Study of Coupling Reaction Using Tetrazole-based Ligand (Sch. Sci., Tokai Univ.) º NAKAMURA, Kaori; KOGUCHI, Shinichi
2G3-20
Oxidation of Alcohol Using IBX-based Ionic Liquid (Sch. Sci., Tokai Univ.) º MIHOYA, Aya; KOGUCHI, Shinichi
Friday, March 27, PM
Chair: ISHIMARU, Yoshihiro
(13:30-14:30)
* 13:20-13:30: interval for laptop PC connection.(2G3-28, 2G3-29, 2G3-30, 2G3-31, 2G3-32, 2G3-33)
2G3-28
NHC-catalyzed reaction, the reactivity of Breslow intermediate in nucleophilic acylation (Grad. Sch. of Sci. Technol., Sophia Univ.; Grad. Sch. Sci., Rikkyo Univ.) º DOBASHI, Kohei; SUZUKI, Yumiko; IWATA, Naoto; ISHITHUBO, Erika; TOKIWA, Hiroaki
2G3-29
Catalytic Aerobic Oxidation of Alcohols by a Mesoionic Derivative (Grad Sch. Eng., Nagoya Inst. of Tech.) º ITO, Satomi; HIRASHITA, Tsunehisa; ARAKI, Shuki
2G3-30
Reactivity of N-Phosphine Oxide-Substituted N-Heterocyclic Carbene (Grad. Sch. Eng., Osaka Univ.) º ASADA, Takahiro; HOSHIMOTO, Yoichi; OHASHI, Masato; SENSUKE, Ogoshi
2G3-31
Synthesis of Novel Thienopyrazines Bearing an Amino Group Using Hypervalent Iodine Reagent and Their Properties (Grad. Sch. Eng., Osaka Univ.) º UETA, Satoshi; TAKEDA, Youhei; MINAKATA, Satoshi
2G3-32
Preparation Conditions of Novel Oligomers Giving Gold-Like Coatings (Grad. Sch. Adv. Integration Sci., Chiba Univ.) º KOBAYASHI, Makoto; MASU, Hyuma; ITOH, Tsutomu; HOSHINO, Katsuyoshi
2G3-33
Synthesis and spectrum of dithenyloxadiazolopyridines emitting FL in NIR region (Grad. Sch. Eng., Kyushu Sangyo Univ.) º IWASAKI, Wataru; NAOMOTO, Kensuke; NAKASHIMA, Takahiro; MATSUOKA, Yohei; YAZUMI, Takashi; KASHIWA, Yuki; NISHI, Kentaro; ISOBE, Shin-ichiro
Chair: HOSHIMOTO, Yoichi
(14:40-15:40)
* 14:30-14:40: interval for laptop PC connection.(2G3-35, 2G3-36, 2G3-37, 2G3-38, 2G3-39, 2G3-40)
2G3-35
Investigation of the steric hindrance factor in antiaromatic porphyrin analog (Grad. Sch. Sci., Eng., Saitama Univ.) º SHIBA, Haruaki; FUJIHARA, Takashi; SETSUNE, Jun-ichiro; ISHIMARU, Yoshihiro
2G3-36
Synthesis and properties of new antiaromatic porphyrin analog containing hetero cycles (Grad. Sch. Sci., Eng., Saitama Univ.) º IKEDA, Ryo; FUJIHARA, Takashi; SETSUNE, Jun-ichiro; ISHIMARU, Yoshihiro
2G3-37
Synthesis and properties of large porphyrinoid compounds with BODIPY (Grad. Sch. Sci., Eng., Saitama Univ.) º TAKAHASHI, Fumiya; FUJIHARA, Takashi; SETSUNE, Jun-ichiro; ISHIMARU, Yoshihiro
2G3-38
Synthesis and properties of Thieno[2,3-d:5,4-d']bisthiazole 4-oxide (Fac. Eng., Gifu Univ.; Fac. Eng., Gifu Univ.) º KAWAI, Yasuhiro; KAGA, Shigesaki; SHIBAHARA, Fumitoshi; MURAI, Toshiaki
2G3-39
Synthesis and evaluation of novel dyes with heterocyclic anchoring group (Yokohama Coll. of Pharmacy; Grad. Sch. Sci., Eng., Tokyo Tech; Grad. Sch. Life Sci. Sys. Eng., KIT) º MASUI, Hisashi; FUSE, Shinichiro; MAITANI, Masato; WADA, Yuji; OGOMI, Yuhei; HAYASE, Shuji; TAKAHASHI, Takashi
2G3-40
Synthesis of novel conjugated phenol derivatives bridged by heterocycles having amyloid-β aggregation inhibitory activity (Grad. Sch. Eng., Iwate Univ.) KAWANO, Tomikazu; º OHASHI, Toshika; OGAWA, Satoshi
Saturday, March 28, AM
Chair: OKAUCHI, Tatsuo
(09:00-10:00)
* 8:50-9:00: interval for laptop PC connection.(3G3-01, 3G3-02, 3G3-03, 3G3-04, 3G3-05, 3G3-06)
3G3-01
Asymmetric Michael/Henry Reaction Using Chiral Bis(imidazolidine)pyridine-Nickel Complex: Synthesis of Novel Chiral Thiochromanyl-Spirooxindole Compounds (Grad. Sch. Sci., Chiba Univ.) º OGAWA, Hiroki; ARAI, Takayoshi
3G3-02
BICMAP-Rhodium Catalyzed Asymmetric 1,4-Addition to Coumarins (Grad. Sch. Eng., Chiba Univ.) MINO, Takashi; º MIURA, Kazuki; MIZUTANI, Yuki; TAGUCHI, Hiroyuki; SAKAMOTO, Masami
3G3-03
Asymmetric Alcohol Addition Reaction Using Isatin-derived Ketimines Catalyzed by Chiral Bis(imidazolidine)pyridine-metal Complex (Grad. Sch. Sci., Chiba Univ.) º TSUCHIYA, Kento; MATSUMURA, Eri; ARAI, Takayoshi
3G3-04
Development of Catalytic Asymmetric Diels-Alder Reaction of Nitro Olefin and Furans Using Chiral Organocatalyst (Grad. Sch. Sci., Osaka City Univ.) º UEDA, Shota; SHINADA, Tetsuro
3G3-05
Synthesis of chiral hydoroxamic acids having pyrroloimidazole structure and their application in asymmetric oxidation (Yokohama Natl. Univ. Engineering Science) º MORITA, Junya; HOSHINO, Yujiro; HONDA, Kiyoshi
3G3-06
The development of multifunctional N-Heterocyclic carbene ligands bearing a pyridine moiety: Copper-catalyzed asymmetric alkylation of N-sulfonylimines with dialkylzinc reagents (Grad. Sch. Nat. Sci. Technol., Kanazawa Univ.) º ISHIZAKA, Tomohiro; SOETA, Takahiro; UKAJI, Yutaka
Chair: SOETA, Takahiro
(10:10-11:10)
* 10:00-10:10: interval for laptop PC connection.(3G3-08, 3G3-09, 3G3-10, 3G3-11, 3G3-12, 3G3-13)
3G3-08
Optical resolution of 2-hydroxymethyltriethylenediamine (Sagami Chemical Research Institute; Grad. Sch. Sci., Kitasato Univ.) º OHTA, Hayato; SHIOSAKI, Masahiro; INOUE, Munenori
3G3-09
Novel Chiral Ionic Liquids Containing hydroxy- or cyano group for Asymmetric Michael Reaction. (Fac. Eng., Oita Univ.) º TANGE, Masakazu; NOBUOKA, Kaoru; KITAOKA, Satoshi; ISHIKAWA, Yuichi
3G3-10
Synthetic Study of Chiral Imidazolium Salts bearing a Bulky Bornane Substituent (Fac. Eng., Iwate Univ.) SHIMADA, Kazuaki; º FUKUMA, Kodai; KORENAGA, Toshinobu
3G3-11
Enantioselective Synthesis of Hetero Helicenes bearing 1,2,3-Triazole units (ISIR, Osaka Univ.) º SAKAI, Tomohiro; YOSHIDA, Yasushi; TAKIZAWA, Shinobu; SASAI, Hiroaki
3G3-12
Novel Chiral Benzimidazole Ligands Having a Spiro Skeleton: Design, Preparation and Application (ISIR, Osaka Univ.) º TAKATANI, Shuhei; SAWADA, Kazuya; TAKENAKA, Kazuhiro; SASAI, Hiroaki
3G3-13
Synthesis and reaction of chiral guanidinodiazonium salt (Grad. Sch. Eng., KIT; Grad. Sch. Eng., KIT) º ISHIKAWA, Akihiro; OKAUCHI, Tatuo; KITAMURA, Mitsuru